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Contents
6
Contributors
10
Pharmacology
11
Introduction
11
Mechanism of Drug Action
12
Pharmacodynamics
18
Pharmacokinetic Principles
23
Introduction
23
Drug Absorption
24
Drug Distribution
29
Drug Metabolism
37
Enzyme Inhibition
41
Drug Excretion (Elimination)
42
Factors Affecting Pharmacokinetics
51
Drug Interactions with a Pharmacokinetic Basis
58
Deciding to Embark on Therapeutic Drug Monitoring
60
Summary
61
Introduction to Specialist Therapeutics
63
Drugs Targeting the Gastrointestinal Tract in Critical Care
63
Sedation on the Intensive Care Unit
67
Nonopioid Analgesia Within the Intensive Care Unit
72
Opiates in Critical Care Introduction
74
Conclusion
76
Index
77
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